Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach

Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach Publisher

Noushini S¹ ; Mahdavi M¹ ; Firoozpour L² ; Moghimi S¹ ; Shafiee A¹ ; Foroumadi A^{1, 2}

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1. Department of Medicinal Chemistry, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran
2. Drug Design and Development Research Center, Tehran University of Medical Sciences, Tehran, Iran

Source: Tetrahedron Published:2015

Abstract

Abstract A new design for the synthesis of 1,2-dihydro-4H-benzo[e][1,4]diazepine-3,5-diones based on Petasis reaction followed by intramolecular amidation in one-pot manner is reported. By employing different primary aromatic and aliphatic amines along with boronic acid derivatives, the desired products have been obtained at ambient temperature in moderate to good yields. © 2015 Elsevier Ltd.

Style	Citing Format
MLA	Noushini S, et al.. "Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach." Tetrahedron, vol. 71, no. 36, 2015, pp. 6272-6275.
APA	Noushini S, Mahdavi M, Firoozpour L, Moghimi S, Shafiee A, Foroumadi A (2015). Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach. Tetrahedron, 71(36), 6272-6275.
Chicago	Noushini S, Mahdavi M, Firoozpour L, Moghimi S, Shafiee A, Foroumadi A. "Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach." Tetrahedron 71, no. 36 (2015): 6272-6275.
Harvard	Noushini S et al. (2015) 'Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach', Tetrahedron, 71(36), pp. 6272-6275.
Vancouver	Noushini S, Mahdavi M, Firoozpour L, Moghimi S, Shafiee A, Foroumadi A. Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach. Tetrahedron. 2015;71(36):6272-6275.
BibTex	@article{ author = {Noushini S and Mahdavi M and Firoozpour L and Moghimi S and Shafiee A and Foroumadi A}, title = {Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach}, journal = {Tetrahedron}, volume = {71}, number = {36}, pages = {6272-6275}, year = {2015} }
RIS	TY - JOUR AU - Noushini S AU - Mahdavi M AU - Firoozpour L AU - Moghimi S AU - Shafiee A AU - Foroumadi A TI - Efficient Multi-Component Synthesis of 1,4-Benzodiazepine-3,5-Diones: A Petasis-Based Approach JO - Tetrahedron VL - 71 IS - 36 SP - 6272 EP - 6275 PY - 2015 ER -

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