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Method for the Synthesis of Chromenopyrimidine-Fused Azoles by Copper-Catalyzed Intramolecular Hetero-Diels–Alder Reaction Publisher



Ghomi MK2 ; Alizadeh N1 ; Moazzam A2 ; Hosseini S3 ; Bahadorikhalili S4 ; Larijani B2 ; Mahdavi M2
Authors

Source: Chemistry of Heterocyclic Compounds Published:2023


Abstract

[Figure not available: see fulltext.] One-pot efficient copper-catalyzed approach for the synthesis of tetracyclic chromeno[4',3':4,5]pyrimido[1,2-b]indazolone and chromeno[4,3-d]-[1,2,4]triazolo[4,3-a]pyrimidine derivatives as a class of pharmacologically interesting compounds through the intramolecular domino condensation–aza-Diels–Alder reaction of aminoazoles and o-propargylated salicylaldehydes under reflux conditions has been described. © 2023, Springer Science+Business Media, LLC, part of Springer Nature.
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