Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles

Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles Publisher

Seifinoferest B¹ ; Tanbakouchian A² ; Larijani B¹ ; Mahdavi M¹

Show Affiliations

1. Endocrinology and Metabolism Research Centre, Tehran University of Medical Sciences, University of Tehran, Nejatollahi St, Enghelab St, Iran
2. Department of Chemistry, College of Chemistry, University of Tehran, 16 Azar St, Enghelab St, Iran

Source: Asian Journal of Organic Chemistry Published:2021

Abstract

The Carbon-Nitrogen bond formation has always been an important and useful tool in drug discovery. Its wide applications in synthesizing N-heterocycles, known as the most prevalent moiety in the active pharmacophores, have attracted increasing attention from researchers. In recent years many works were devoted to finding new and more rapid and effective chemo- and regio-selective methods for the synthesis of N-containing heterocycles. Buchwald-Hartwig and Ullman-Goldberg are two proven efficient methods for synthesizing five, six, and seven-membered heterocycles found abundantly in literature. Here, we study these two amination methods more precisely, based on the reaction conditions and the products. © 2021 Wiley-VCH GmbH

Style	Citing Format
MLA	Seifinoferest B, et al.. "Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles." Asian Journal of Organic Chemistry, vol. 10, no. 6, 2021, pp. 1319-1344.
APA	Seifinoferest B, Tanbakouchian A, Larijani B, Mahdavi M (2021). Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles. Asian Journal of Organic Chemistry, 10(6), 1319-1344.
Chicago	Seifinoferest B, Tanbakouchian A, Larijani B, Mahdavi M. "Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles." Asian Journal of Organic Chemistry 10, no. 6 (2021): 1319-1344.
Harvard	Seifinoferest B et al. (2021) 'Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles', Asian Journal of Organic Chemistry, 10(6), pp. 1319-1344.
Vancouver	Seifinoferest B, Tanbakouchian A, Larijani B, Mahdavi M. Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles. Asian Journal of Organic Chemistry. 2021;10(6):1319-1344.
BibTex	@article{ author = {Seifinoferest B and Tanbakouchian A and Larijani B and Mahdavi M}, title = {Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles}, journal = {Asian Journal of Organic Chemistry}, volume = {10}, number = {6}, pages = {1319-1344}, year = {2021} }
RIS	TY - JOUR AU - Seifinoferest B AU - Tanbakouchian A AU - Larijani B AU - Mahdavi M TI - Ullmann-Goldberg and Buchwald-Hartwig C−N Cross Couplings: Synthetic Methods to Pharmaceutically Potential N-Heterocycles JO - Asian Journal of Organic Chemistry VL - 10 IS - 6 SP - 1319 EP - 1344 PY - 2021 ER -

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