Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives

Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives Publisher

Mahdavi M¹ ; Bialam M² ; Saeedi M³ ; Jafarpour F² ; Foroumadi A¹ ; Shafiee A¹

Show Affiliations

1. Department of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, 14176, Iran
2. School of Chemistry, College of Science, University of Tehran, PO Box 14155-6455, Tehran, Iran
3. Persian Medicine and Pharmacy Research Center, Tehran University of Medical Sciences, Tehran, Iran

Source: Synlett Published:2015

Abstract

Substituted o-Amino-N-(prop-2-yn-1-yl) aromatic amides easily reacted with carbon disulfide (CS2) in the presence of potassium hydroxide (KOH) in EtOH under reflux conditions. Cyclization reaction followed by a favored 5-exo-dig ring closure afforded 2-methylene-thiazolo[2,3-b]quinazolinone derivatives in good yields. © Georg Thieme Verlag Stuttgart New York.

Style	Citing Format
MLA	Mahdavi M, et al.. "Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives." Synlett, vol. 26, no. 2, 2015, pp. 173-176.
APA	Mahdavi M, Bialam M, Saeedi M, Jafarpour F, Foroumadi A, Shafiee A (2015). Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives. Synlett, 26(2), 173-176.
Chicago	Mahdavi M, Bialam M, Saeedi M, Jafarpour F, Foroumadi A, Shafiee A. "Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives." Synlett 26, no. 2 (2015): 173-176.
Harvard	Mahdavi M et al. (2015) 'Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives', Synlett, 26(2), pp. 173-176.
Vancouver	Mahdavi M, Bialam M, Saeedi M, Jafarpour F, Foroumadi A, Shafiee A. Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives. Synlett. 2015;26(2):173-176.
BibTex	@article{ author = {Mahdavi M and Bialam M and Saeedi M and Jafarpour F and Foroumadi A and Shafiee A}, title = {Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives}, journal = {Synlett}, volume = {26}, number = {2}, pages = {173-176}, year = {2015} }
RIS	TY - JOUR AU - Mahdavi M AU - Bialam M AU - Saeedi M AU - Jafarpour F AU - Foroumadi A AU - Shafiee A TI - Efficient Synthesis of 2-Methylenethiazolo[2,3- B ]Quinazolinone Derivatives JO - Synlett VL - 26 IS - 2 SP - 173 EP - 176 PY - 2015 ER -

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