Tehran University of Medical Sciences

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Faculty Members have conducted research related to the Novel 5-Fluoro-6-(4-(2-Fluorophenyl)Piperazin-1-Yl)-2-(4-(4-Methylpiperazin-1-Yl)Phenyl)-1H-Benzo[D]Imidazole Derivatives As Promising Urease Inhib-Itors
Mohsen Amini
Mohsen Amini

Professor of Pharmaceutical Chemistry

Department Medicinal Chemistry

School of Pharmacy

Drug Design and Development Research Center

Tehran University of Medical Sciences

All Documents
1. A Comprehensive Review on the Latest Advances of Dimeric Anticancer Prodrugs, Future Medicinal Chemistry (2025)
2. Comprehensive Analysis of Bioactive Compounds in Malt Beverages: A Chemometric Approach for Quality Control, Journal of Agricultural Science and Technology (2025)
3. Design, Synthesis, and Investigation of Novel 5-Arylpyrazole-Glucose Hybrids As Α-Glucosidase Inhibitors, Scientific Reports (2025)
4. Design, Synthesis, Anticonvulsant Evaluation, and Molecular Docking Studies of New Gabaa Agonist Derivatives, Iranian Journal of Pharmaceutical Research (2025)
5. In the Pursuit of an Efficient Delignification From Pumpkin Seed Shells by the Polyextremophilic and Laccase-Producing Bacterial Isolate Halomonas Elongata, Biomass Conversion and Biorefinery (2025)
6. Metal-Organic Frameworks Mil-101(Fe) and Mil-53(Al) As Efficient Adsorbents for Dispersive Micro-Solid-Phase Extraction of Sorafenib in Plasma and Wastewater, Coupled With Hplc-Uv Analysis, Journal of Chromatographic Science (2025)
7. The Most Up-To-Date Advancements in the Design and Development of Urease Inhibitors (January 2020-March 2024), Journal of Agricultural and Food Chemistry (2025)
8. A Gc-Ms Method for Determination of Β-Propiolactone Residues in Inactivated Covid-19 Vaccines, Journal of Chromatographic Science (2024)
9. A Novel Ph-Sensitive Nanocomposite Based on Graphene Oxide for Improving Doxorubicin Release, Current Drug Delivery (2024)
10. A Review on Zinc, Cadmium, and Mercury Complexes With Anticancer Activity, Inorganic Chemistry Communications (2024)
11. Comparative Study of Dispersive Micro-Solid Phase Extraction of Nandrolone Using Mil-53(Al) and Zif-8 in Human Plasma, Journal of Analytical Chemistry (2024)
12. Comparison of Testosterone Extraction From Human Plasma Using Mofs (Mil-53(Al) and Zif-8)-Based D-Μ-Spe Coupled to Hplc–Uv, Chromatographia (2024)
13. Development of a High-Performance Liquid Chromatography Using Rhodamine B Hydrazide As the Derivatization Reagent for Determination of Β Propiolactone Residues in Inactivated Covid-19 Vaccines, Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences (2024)
14. Development of Non-Destructive Methods for the Assessment of Authenticity of Sports Whey Protein Supplements, Food Additives and Contaminants - Part A (2024)
15. Development, Optimization, and Characterization of Vitamin C-Fortified Oleogel-Based Chewable Gels and a Novel Nondestructive Analysis Method for the Vitamin C Assay, Food Production, Processing and Nutrition (2024)
16. Dispersive Micro-Solid Phase Extraction Based on Two Mofs As Highly Effective Adsorbents for Analysis of Nilotinib in Plasma and Wastewater, DARU, Journal of Pharmaceutical Sciences (2024)
17. Enzymatic Dual-Faced Janus Structures Based on the Hierarchical Organic-Inorganic Hybrid Matrix for an Effective Bioremoval and Detoxification of Reactive Blue-19, International Journal of Biological Macromolecules (2024)
18. Forced Degradation Products of Liraglutide: A Comparative Study of Similarity Between Originator and Analogue Version by Liquid Chromatography–Mass Spectrometry, International Journal of Peptide Research and Therapeutics (2024)
19. Novel 5-Fluoro-6-(4-(2-Fluorophenyl)Piperazin-1-Yl)-2-(4-(4-Methylpiperazin-1-Yl)Phenyl)-1H-Benzo[D]Imidazole Derivatives As Promising Urease Inhib-Itors, Letters in Drug Design and Discovery (2024)
20. Pegylated Mesoporous Silica Core–Shell Redox-Responsive Nanoparticles for Delivering Paclitaxel to Breast Cancer Cells, International Journal of Pharmaceutics (2024)
21. Preparation of Novel 3,4,5-Triaryl-1,2,4-Oxadiazole Derivatives: Molecular Docking and Α-Glucosidase Assessment, ChemistrySelect (2024)
22. Preparation, Characterization and in Vitro Evaluation of Insulin-Phbv Nanoparticles/Alginate Hydrogel Composite System for Prolonged Delivery of Insulin, Journal of Pharmaceutical Sciences (2024)
23. Recent Advances in Design and Development of Diazole and Diazine Based Fungicides (2014-2023), Journal of Agricultural and Food Chemistry (2024)
24. Salvia Mirzayanii and Salvia Hypoleuca Essential Oils: Chemical Composition, Alpha-Glucosidase Inhibitory, and Synergistic Effects of Selected Components, Jundishapur Journal of Natural Pharmaceutical Products (2024)
25. Synthesis and in Silico Admet Evaluation of New Thiazole and Thiazolidine-4-One Derivatives As Non-Ulcerogenic Analgesic and Anti-Inflammatory Agents, Journal of the Serbian Chemical Society (2024)
26. Synthesis, Biological Evaluation, and in Silico Study of Novel Coumarin-Quinazoline Analogs As Potential Anti-Angiogenesis Agents, Results in Chemistry (2024)
27. Targeted Ph- and Redox-Responsive Aus/Micelles With Low Cmc for Highly Efficient Sonodynamic Therapy of Metastatic Breast Cancer, Biomaterials Advances (2024)
28. 2-Aryl Benzimidazole Derivatives Act As Potent Urease Inhibitors; Synthesis, Bioactivity and Molecular Docking Study, Polycyclic Aromatic Compounds (2023)
29. Biological Activity of Novel Pyrrole Derivatives As Antioxidant Agents Against 6-Ohda Induced Neurotoxicity in Pc12 Cells, Iranian Journal of Pharmaceutical Research (2023)
30. Corrigendum to “Dual Drug Delivery System of Plga Nanoparticles to Reverse Drug Resistance by Altering Bax/Bcl-2” [J. Drug Deliv. Sci. Technol. 47 (2018) 291–298, (S1773224718301825), (10.1016/J.Jddst.2018.07.019)], Journal of Drug Delivery Science and Technology (2023)
31. Fabrication, Characterization and Evaluation of a New Designed Botulinum Toxin-Cell Penetrating Peptide Nanoparticulate Complex, DARU# Journal of Pharmaceutical Sciences (2023)
32. New Bioactive Dipiperazine Derivatives; Synthesis, Molecular Docking and Urease Inhibition Study, ChemistrySelect (2023)
33. New Imidazo[1,2-A]Pyridin-2-Yl Derivatives As Ache, Bche, and Lox Inhibitors; Design, Synthesis, and Biological Evaluation, Letters in Drug Design and Discovery (2023)
34. Preparation of Polymersomes From Synthesized Hyaluronic Acid-Graft-Poly(Ε-Caprolactone) Copolymers for Drug Delivery to the Brain, Materials Today Chemistry (2023)
35. Rapid Determination of Ethanol in Non-Alcoholic Malt Beverage by Atr-Ft-Ir Spectroscopy and Headspace Gas Chromatography Confirmation, Journal of Agricultural Science and Technology (2023)
36. Simultaneous Extraction of Six Phthalic Acid Esters From Polyethylene Terephthalate (Pet) Bottled Water Using Poly (Ionic Liquid) Functionalised Silica Coated-Iron Oxide Nanoparticles: A Risk Assessment Study, International Journal of Environmental Analytical Chemistry (2023)
37. Synthesis, Bioactivity, and Molecular Docking of Benzimidazole-2-Carbamate Derivatives As Potent Α-Glucosidase Inhibitors, Journal of Molecular Structure (2023)
38. Synthesis, Docking Study, and Biological Evaluation of 2-Phenylchroman-4-One Derivatives As Murine Double Minute 2 (Mdm2) Inhibitors, ChemistrySelect (2023)
39. Thioquinoline Derivatives Conjugated to Thiosemicarbazide As Potent Tyrosinase Inhibitors With Anti-Melanogenesis Properties, Scientific Reports (2023)
40. An Approach to Pharmacological Targets of Pyrrole Family From Medicinal Chemistry Viewpoint, Mini-Reviews in Medicinal Chemistry (2022)
41. Benzimidazole Derivatives Act As Dual Urease Inhibitor and Anti-Helicobacter Pylori Agent; Synthesis, Bioactivity, and Molecular Docking Study, Synthetic Communications (2022)
42. Design, Synthesis, and Bioactivity Investigation of Novel Benzimidazole Derivatives As Potent Urease Inhibitors, Synthetic Communications (2022)
43. Evaluation of Dna Methylation in Bdnf, Slc6a4, Nr3c1 and Fkbp5 Before and After Treatment With Selective Serotonin-Reuptake Inhibitor in Major Depressive Disorder, Epigenomics (2022)
44. Fatty Acid Composition of Iranian Sweetened Confectionery Creams, With an Emphasis on Trans Fatty Acids, Journal of Food Composition and Analysis (2022)
45. Influence of Cooking Process on the Content of Water-Soluble B Vitamins in Rice Marketed in Iran, Food Science and Nutrition (2022)
46. Novel Benzimidazole Derivatives; Synthesis, Bioactivity and Molecular Docking Study As Potent Urease Inhibitors, DARU# Journal of Pharmaceutical Sciences (2022)
47. Piperazine-Based Semicarbazone Derivatives As Potent Urease Inhibitors: Design, Synthesis, and Bioactivity Screening, Letters in Drug Design and Discovery (2022)
48. Synthesis and Biological Evaluation of Novel Anti-Leukemia Proteolysis-Targeting Chimeras in Degradating Inosine Monophosphate Dehydrogenase, Iranian Journal of Pharmaceutical Research (2022)
49. Synthesis, Molecular Docking and Biological Evaluation of Diaryl Pyrimidine Derivatives As Urease Inhibitors, Pharmaceutical Chemistry Journal (2022)
50. Synthesis, Molecular Docking, and Biological Evaluation of 2,3-Diphenylquinoxaline Derivatives As a Tubulin’S Colchicine Binding Site Inhibitor Based on Primary Virtual Screening, Anti-Cancer Agents in Medicinal Chemistry (2022)
51. Thiosemicarbazone Derivatives Act As Potent Urease Inhibitors; Synthesis, Bioactivity Screening and Molecular Docking Study, ChemistrySelect (2022)
52. 5-Benzylidene-2,3-Diarylthiazolidine-4-Ones: Design, Synthesis, Spectroscopic Characterization, in Vitro Biological and Computational Evaluation, Synthetic Communications (2021)
53. Changes in Dna Methylation in Apoe and Ackr3 Genes in Multiple Sclerosis Patients and the Relationship With Their Heavy Metal Blood Levels, NeuroToxicology (2021)
54. Changes in Dna Methylation in Apoe and Ackr3 Genes in Multiple Sclerosis Patients and the Relationship With Their Heavy Metal Blood Levels, NeuroToxicology (2021)
55. Design, Synthesis and Bioactivity Investigation of Novel 2,3-Diarylthiazolidine-4-Ones As Potent Α-Glucosidase Inhibitors, Polycyclic Aromatic Compounds (2021)
56. Design, Synthesis, Andin Vitroandin Vivoevaluation of Novel Fluconazole-Based Compounds With Promising Antifungal Activities, ACS Omega (2021)
57. Developing Novel Anticancer Drugs for Targeted Populations: An Update, Current Pharmaceutical Design (2021)
58. Glutamate-Urea-Based Psma-Targeted Plga Nanoparticles for Prostate Cancer Delivery of Docetaxel, Pharmaceutical Development and Technology (2021)
59. Novel Combined Topical Gel of Lidocaine–Verapamil–Nitroglycerin Can Dilate the Radial Artery and Reduce Radial Pain During Trans-Radial Angioplasty, IJC Heart and Vasculature (2021)
60. Optimization of the Culture Medium and Characterization of Antioxidant Compounds of a Marine Isolated Microalga As a Promising Source in Aquaculture Feed, Biocatalysis and Agricultural Biotechnology (2021)
61. Preparation and Pulsatile Release Evaluation of Teriparatide-Loaded Multilayer Implant Composed of Polyanhydride-Hydrogel Layers Using Spin Coating for the Treatment of Osteoporosis, Journal of Pharmaceutical Innovation (2021)
62. Pyrazole Derivatives Induce Apoptosis Via Ros Generation in the Triple Negative Breast Cancer Cells, Mda-Mb-468, Asian Pacific Journal of Cancer Prevention (2021)
63. Study on the Interaction of 1,5-Diaryl Pyrrole Derivatives With Αglucosidase; Synthesis, Molecular Docking, and Kinetic Study, Medicinal Chemistry (2021)
64. Synthesis, Biological Evaluation and Docking Study of New Pyrimidine Compounds As Anticancer Agents, Drug Research (2021)
65. Synthesis, Evaluation of Biological Activity, Docking and Molecular Dynamic Studies of Pyrimidine Derivatives, Letters in Organic Chemistry (2021)
66. Triarylpyrazole Derivatives As Potent Cytotoxic Agents; Synthesis and Bioactivity Evaluation Pyrazole Derivatives As Anticancer Agent, Drug Research (2021)
67. Anticholinesterase Activity of Cinnamic Acids Derivatives: In Vitro, in Vivo Biological Evaluation, and Docking Study, Letters in Drug Design and Discovery (2020)
68. Cadmium Accumulation and Alkaloid Production of Narcissus Tazetta Plants Grown Under in Vitro Condition With Cadmium Stress, Plant Physiology Reports (2020)
69. Co-Delivery of Gemcitabine Prodrug Along With Anti Nf-Κb Sirna by Tri-Layer Micelles Can Increase Cytotoxicity, Uptake and Accumulation of the System in the Cancers, Materials Science and Engineering C (2020)
70. Combining Chemometrics and the Technique for the Order of Preference by Similarity to Ideal Solution: A New Approach to Multiple-Response Optimization of Hplc Compared to Desirability Function, Microchemical Journal (2020)
71. Coumarin-Based Scaffold As Α-Glucosidase Inhibitory Activity: Implication for the Development of Potent Antidiabetic Agents, Mini-Reviews in Medicinal Chemistry (2020)
72. Design and Fabrication of Dual-Targeted Delivery System Based on Gemcitabine-Conjugated Human Serum Albumin Nanoparticles, Chemical Biology and Drug Design (2020)
73. Design, Preparation and Biological Evaluation of a 177Lu-Labeled Somatostatin Receptor Antagonist for Targeted Therapy of Neuroendocrine Tumors, Bioorganic Chemistry (2020)
74. Design, Synthesis and Biological Evaluation of Novel Diaryl Pyrazole Derivatives As Anticancer Agents, Letters in Organic Chemistry (2020)
75. Design, Synthesis and In-Vitro Anti-Cancer Evaluation of Novel Derivatives of 2-(2-Methyl-1,5-Diaryl-1H-Pyrrol-3-Yl)-2-Oxo-N-(Pyridin-3-Yl)Acetamide, Medicinal Chemistry (2020)
76. Design, Synthesis, and Evaluation of Novel Cinnamic Acid-Tryptamine Hybrid for Inhibition of Acetylcholinesterase and Butyrylcholinesterase, DARU# Journal of Pharmaceutical Sciences (2020)
77. Design, Synthesis, in Vivo and in Vitro Studies of 1,2,3,4-Tetrahydro-9H-Carbazole Derivatives, Highly Selective and Potent Butyrylcholinesterase Inhibitors, Molecular Diversity (2020)
78. Design, Synthesis, Radiolabeling and Biological Evaluation of New Urea-Based Peptides Targeting Prostate Specific Membrane Antigen, Bioorganic Chemistry (2020)
79. Enzyme Inhibition, Kinetic, and Molecular Docking Studies of Α-Glucosidase, Current Enzyme Inhibition (2020)
80. Hydroxypropyl Beta Cyclodextrin: A Water-Replacement Agent or a Surfactant Upon Spray Freeze-Drying of Igg With Enhanced Stability and Aerosolization, Drug Development and Industrial Pharmacy (2020)
81. Improving the In-Vivo Biological Activity of Fingolimod Loaded Phbv Nanoparticles by Using Hydrophobically Modified Alginate, Drug Development and Industrial Pharmacy (2020)
82. Mitochondrial Delivery of Microrna Mimic Let-7B to Nsclc Cells by Pamam-Based Nanoparticles, Journal of Drug Targeting (2020)
83. Nanofibrous Scaffolds Containing Hydroxyapatite and Microfluidic-Prepared Polyamidoamin/Bmp-2 Plasmid Dendriplexes for Bone Tissue Engineering Applications, International Journal of Nanomedicine (2020)
84. Peg1000 As a Low Melting and Ecofriendly Solvent for Air Oxidative and Catalyst Free 2,4-Disubstitute Quinazoline Synthesis, Letters in Organic Chemistry (2020)
85. Preclinical Study of a New 177Lu-Labeled Somatostatin Receptor Antagonist in Ht-29 Human Colorectal Cancer Cells, Asia Oceania Journal of Nuclear Medicine and Biology (2020)
86. Preparation and Characterization of Albumin Nanoparticles of Paclitaxel-Triphenylphosphonium Conjugates: New Approach to Subcellular Targeting, Drug research (2020)
87. Synthesis and Biological Evaluation of 2-(2-Methyl-1H-Pyrrol-3-Yl)-2-Oxo-N-(Pyridine-3-Yl) Acetamide Derivatives: In Vitro Α-Glucosidase Inhibition, and Kinetic and Molecular Docking Study, Chemical Papers (2020)
88. Synthesis, Biological Evaluation and Preclinical Study of a Novel 99Mtc-Peptide: A Targeting Probe of Amyloid-Β Plaques As a Possible Diagnostic Agent for Alzheimer's Disease, Bioorganic Chemistry (2020)
89. Synthesis, Molecular Docking and Α-Glucosidase Inhibitory Activity Study of 2,4,6-Triaryl Pyrimidine Derivatives, Letters in Drug Design and Discovery (2020)
90. The Antidiabetic and Antilipidemic Effects of Hibiscus Sabdariffa: A Systematic Review and Meta-Analysis of Randomized Clinical Trials, Food Research International (2020)
91. The Antidiabetic Effect of Thymoquinone: A Systematic Review and Meta-Analysis of Animal Studies, Food Research International (2020)
92. Two Novel Anticancer Compounds With Minimum Cardiotoxic Property, BMC Pharmacology and Toxicology (2020)
93. Two Novel Compounds With Tri-Aryl Structures As Effectivanti-Breast Cancer Candidates In-Vivo, Iranian Journal of Pharmaceutical Research (2020)
94. 2,4-Disubstituted Quinazoline Derivatives Act As Inducers of Tubulin Polymerization: Synthesis and Cytotoxicity, Anti-Cancer Agents in Medicinal Chemistry (2019)
95. Anticancer Properties of N-Alkyl-2, 4-Diphenylimidazo [1, 2-A] Quinoxalin-1-Amine Derivatives; Kinase Inhibitors, Bioorganic Chemistry (2019)
96. Antidiabetic Effect of Quercetin: A Systematic Review and Meta-Analysis of Animal Studies, Food and Chemical Toxicology (2019)
97. Design, Synthesis and Anticancer Evaluation of Novel Series of Indibulin Analogues, Medicinal Chemistry (2019)
98. Design, Synthesis, Radiolabeling, and Biologic Evaluation of Three 18F-Fdg-Radiolabeled Targeting Peptides for the Imaging of Apoptosis, Cancer Biotherapy and Radiopharmaceuticals (2019)
99. Development of Octreotide-Loaded Chitosan and Heparin Nanoparticles: Evaluation of Surface Modification Effect on Physicochemical Properties and Macrophage Uptake, Journal of Pharmaceutical Sciences (2019)
100. Enhancement Mitochondrial Apoptosis in Breast Cancer Cells by Paclitaxel-Triphenylphosphonium Conjugate in Dna Aptamer Modified Nanoparticles, Journal of Drug Delivery Science and Technology (2019)
101. Inhibiting Hepatic Gluconeogenesis by Chitosan Lactate Nanoparticles Containing Crtc2 Sirna Targeted by Poly(Ethylene Glycol)-Glycyrrhetinic Acid, Drug Delivery and Translational Research (2019)
102. New Folate Receptor Targeted Nano Liposomes for Delivery of 5-Fluorouracil to Cancer Cells: Strong Implication for Enhanced Potency and Safety, Life Sciences (2019)
103. Novel Morpholine Containing Cinnamoyl Amides As Potent Tyrosinase Inhibitors, International Journal of Biological Macromolecules (2019)
104. Oliveria Decumbens, a Bioactive Essential Oil: Chemical Composition and Biological Activities, Iranian Journal of Pharmaceutical Research (2019)
105. Preparation of Magnetic Iron Oxide Nanoparticles Modified With Imidazolium-Based Ionic Liquids As a Sorbent for the Extraction of Eight Phthalate Acid Esters in Water Samples Followed by Uplc-Ms/Ms Analysis: An Experimental Design Methodology, Analytical Methods (2019)
106. Production of Vitamin D3 Enriched Biomass of Saccharomyces Cerevisiae As a Potential Food Supplement: Evaluation and Optimization of Culture Conditions Using Plackett–Burman and Response Surface Methodological Approaches, Iranian Journal of Pharmaceutical Research (2019)
107. Simultaneous Determination of Nine Sunscreen Agents by Hplc and Chemometric Analysis, Journal of Cosmetic Science (2019)
108. Synthesis and Anti-Breast Cancer Activity of Novel Indibulin Related Diarylpyrrole Derivatives, DARU# Journal of Pharmaceutical Sciences (2019)
109. Synthesis, Anti-Proliferative Evaluation, and Molecular Docking Studies of 3-(Alkylthio)-5,6-Diaryl-1,2,4-Triazines As Tubulin Polymerization Inhibitors, Letters in Drug Design and Discovery (2019)
110. Thiolated Chitosan-Lauric Acid As a New Chitosan Derivative: Synthesis, Characterization and Cytotoxicity, International Journal of Biological Macromolecules (2019)
111. Two Novel Tri-Aryl Derivatives Attenuate the Invasion-Promoting Effects of Stromal Mesenchymal Stem Cells on Breast Cancer, Anti-Cancer Agents in Medicinal Chemistry (2019)
112. 2-[2-Methyl-5-Phenyl-1-(3,4,5-Trimethoxyphenyl)-1Hpyrrol- 3-Yl]-2-Oxo-N-(Pyridin-4-Yl) Acetamide, MolBank (2018)
113. A Magnetic Heterogeneous Biocatalyst Composed of Immobilized Laccase and 2,2,6,6-Tetramethylpiperidine-1-Oxyl (Tempo) for Green One-Pot Cascade Synthesis of 2-Substituted Benzimidazole and Benzoxazole Derivatives Under Mild Reaction Conditions, Advanced Synthesis and Catalysis (2018)
114. A Mechanistic Study of the Effect of Transferrin Conjugation on Cytotoxicity of Targeted Liposomes, Journal of Microencapsulation (2018)
115. A Novel 5-Fluorouracil Targeted Delivery to Colon Cancer Using Folic Acid Conjugated Liposomes, Biomedicine and Pharmacotherapy (2018)
116. Alteration of Hepatocellular Antioxidant Gene Expression Pattern and Biomarkers of Oxidative Damage in Diazinon-Induced Acute Toxicity in Wistar Rat: A Time–Course Mechanistic Study, EXCLI Journal (2018)
117. Characterization of Folic Acid Surface-Coated Selenium Nanoparticles and Corresponding in Vitro and in Vivo Effects Against Breast Cancer, Archives of Medical Research (2018)
118. Co-Immobilization of Laccase and Tempo in the Compartments of Mesoporous Silica for a Green and One-Pot Cascade Synthesis of Coumarins by Knoevenagel Condensation, ChemCatChem (2018)
119. Consistency Evaluation Between Matrix Components Ratio and Microbiological Potency of Tylosin Major Components, DARU# Journal of Pharmaceutical Sciences (2018)
120. Design, Synthesis and Cytotoxicity Evaluation of Indibulin Analogs, Heterocyclic Communications (2018)
121. Design, Synthesis, and Biological Evaluation of Selective and Potent Carbazole-Based Butyrylcholinesterase Inhibitors, Bioorganic and Medicinal Chemistry (2018)
122. Dual Drug Delivery System of Plga Nanoparticles to Reverse Drug Resistance by Altering Bax/Bcl-2, Journal of Drug Delivery Science and Technology (2018)
123. Effects of Coating Layer and Release Medium on Release Profile From Coated Capsules With Eudragit Fs 30D: An in Vitro and in Vivo Study, Drug Development and Industrial Pharmacy (2018)
124. Folic Acid-Modified Liposomal Drug Delivery Strategy for Tumor Targeting of 5-Fluorouracil, European Journal of Pharmaceutical Sciences (2018)
125. Gas Chromatography–Mass Spectrometry Determination of Pregabalin in Human Plasma Using Derivatization Method, Chromatographia (2018)
126. Glutathione Responsive Chitosan-Thiolated Dextran Conjugated Mir-145 Nanoparticles Targeted With As1411 Aptamer for Cancer Treatment, Carbohydrate Polymers (2018)
127. In Vivo Evaluation of Ph and Time-Dependent Polymers As Coating Agent for Colonic Delivery Using Central Composite Design, Journal of Drug Delivery Science and Technology (2018)
128. Luteolin Reduced the Traumatic Brain Injury-Induced Memory Impairments in Rats: Attenuating Oxidative Stress and Dark Neurons of Hippocampus, Acta Medica Iranica (2018)
129. Novel and Efficient Method for Solid Phase Synthesis of Urea-Containing Peptides Targeting Prostate Specific Membrane Antigen (Psma) in Comparison With Current Methods, Iranian Journal of Pharmaceutical Research (2018)
130. Novel Cinnamic Acid–Tryptamine Hybrids As Potent Butyrylcholinesterase Inhibitors: Synthesis, Biological Evaluation, and Docking Study, Archiv der Pharmazie (2018)
131. Novel Tetrahydrocarbazole Benzyl Pyridine Hybrids As Potent and Selective Butryl Cholinesterase Inhibitors With Neuroprotective and Β-Secretase Inhibition Activities, European Journal of Medicinal Chemistry (2018)
132. Synthesis and Characterization of a Novel Peptide-Grafted Cs and Evaluation of Its Nanoparticles for the Oral Delivery of Insulin, in Vitro, and in Vivo Study, International Journal of Nanomedicine (2018)
133. Synthesis and Characterization of Novel Phthalimide-Pyrano[3,2-C]Chromene and Phthalimide-Pyrano-2-One Hybrids, Journal of Heterocyclic Chemistry (2018)
134. Transferrin Targeted Liposomal 5-Fluorouracil Induced Apoptosis Via Mitochondria Signaling Pathway in Cancer Cells, Life Sciences (2018)
135. A Novel Nanoemulsion-Based Method to Produce Ultrasmall, Water-Dispersible Nanoparticles From Chitosan, Surface Modified With Cell-Penetrating Peptide for Oral Delivery of Proteins and Peptides, International Journal of Nanomedicine (2017)
136. Anticonvulsant Effects of New 1, 4-Dihydropyridinederivatives Containing Imidazolyl Moiety Against Seizures Induced by Pentylenetetrazole and Maximal Electroshock in Mice, Iranian Journal of Pharmaceutical Research (2017)
137. Application of Artificial Neural Networks in the Design and Optimization of a Nanoparticulate Fingolimod Delivery System Based on Biodegradable Poly(3-Hydroxybutyrate-Co-3-Hydroxyvalerate), Journal of Pharmaceutical Sciences (2017)
138. Biotin Decorated Plga Nanoparticles Containing Sn-38 Designed for Cancer Therapy, Artificial Cells# Nanomedicine and Biotechnology (2017)
139. Development of an Rp-Hplc-Uv Method for Simultaneous Detection of Nimodipine and Its Metabolite in Cerebrospinal Fluid of Rat, Iranian Journal of Pharmaceutical Research (2017)
140. In-Vitro Cytotoxicity and Combination Effects of the Docetaxel-Conjugated and Doxorubicin-Conjugated Poly(Lactic Acid)-Poly(Ethylene Glycol)-Folate-Based Polymeric Micelles in Human Ovarian Cancer Cells, Journal of Pharmacy and Pharmacology (2017)
141. Ion-Pair Switchable-Hydrophilicity Solvent-Based Homogeneous Liquid–Liquid Microextraction for the Determination of Paraquat in Environmental and Biological Samples Before High-Performance Liquid Chromatography, Journal of Separation Science (2017)
142. Nano Polyelectrolyte Complexes of Carboxymethyl Dextran and Chitosan to Improve Chitosan-Mediated Delivery of Mir-145, Carbohydrate Polymers (2017)
143. Novel 4-Thiazolidinone Derivatives As Agonists of Benzodiazepine Receptors: Design, Synthesis and Pharmacological Evaluation, EXCLI Journal (2017)
144. Optimization of Culture Conditions for Enrichment of Saccharomyces Cerevisiae With Dl-Α-Tocopherol by Response Surface Methodology, Iranian Journal of Pharmaceutical Research (2017)
145. Peptide Functionalized Poly Ethylene Glycol-Poly Caprolactone Nanomicelles for Specific Cabazitaxel Delivery to Metastatic Breast Cancer Cells, Materials Science and Engineering C (2017)
146. Preparation of Human Serum Albumin Nanoparticles Using a Chemometric Technique, Journal of Nanostructure in Chemistry (2017)
147. Preparation, Characterization and in Vivo Evaluation of a Combination Delivery System Based on Hyaluronic Acid/Jeffamine Hydrogel Loaded With Phbv/Plga Blend Nanoparticles for Prolonged Delivery of Teriparatide, European Journal of Pharmaceutical Sciences (2017)
148. Rapid Analysis of Styrene in Drinking Water and Tea Samples Using Dispersive Liquid-Liquid Microextraction Combined With Liquid Chromatography-Ultraviolet Detection, Food Analytical Methods (2017)
149. Simultaneous Determination of Preservatives in Dairy Products by Hplc and Chemometric Analysis, International Journal of Analytical Chemistry (2017)
150. Solid Lipid Nanoparticles Surface Modified With Anti-Contactin-2 or Anti-Neurofascin for Brain-Targeted Delivery of Medicines, Pharmaceutical Development and Technology (2017)
151. Synthesis and Neuroprotective Activity of Novel 1,2,4-Triazine Derivatives With Ethyl Acetate Moiety Against H2o2 and Aβ-Induced Neurotoxicity, Medicinal Chemistry Research (2017)
152. Synthesis of (2-Mercaptoacetyl)-L-[2-14C]Tryptophan As a Selective Metallo-Β-Lactamase Inhibitor Via [2-14C]Indole Based on Chiral Pool Strategy, Journal of Labelled Compounds and Radiopharmaceuticals (2017)
153. Synthesis, Docking Study and Neuroprotective Effects of Some Novel Pyrano[3,2-C]Chromene Derivatives Bearing Morpholine/Phenylpiperazine Moiety, Bioorganic and Medicinal Chemistry (2017)
154. Targeted Delivery of Cabazitaxel by Conjugation to Albumin-Peg-Folate Nanoparticles Using a Cysteine-Acrylate Linker and Simple Synthesis Conditions, Current Drug Delivery (2017)
155. Targeted Dna Delivery to Cancer Cells Using a Biotinylated Chitosan Carrier, Biotechnology and Applied Biochemistry (2017)
156. The Effect of Freeze-Dried Antibody Concentrations on Its Stability in the Presence of Trehalose and Hydroxypropyl-Β-Cyclodextrin: A Box–Behnken Statistical Design, Pharmaceutical Development and Technology (2017)
157. Ultrasonic Assisted Switchable Solvent Based on Liquid Phase Microextraction Combined With Micro Sample Injection Flame Atomic Absorption Spectrometry for Determination of Some Heavy Metals in Water, Urine and Tea Infusion Samples, Journal of Molecular Liquids (2017)
158. 18Fdg-Labeled Likkpf: A Pet Tracer for Apoptosis Imaging, Journal of Radioanalytical and Nuclear Chemistry (2016)
159. Biotin/Folate-Decorated Human Serum Albumin Nanoparticles of Docetaxel: Comparison of Chemically Conjugated Nanostructures and Physically Loaded Nanoparticles for Targeting of Breast Cancer, Chemical Biology and Drug Design (2016)
160. Design, Synthesis and Anti-Tubercular Activity of Novel 1, 4-Dihydropyrine-3, 5-Dicarboxamide Containing 4(5)-Chloro-2-Ethyl-5(4)-Imidazolyl Moiety, Iranian Journal of Pharmaceutical Research (2016)
161. Design, Synthesis and Evaluation of New Azoles As Antifungal Agents: A Molecular Hybridization Approach, Pharmaceutical Chemistry Journal (2016)
162. Development of Molecularly Imprinted Olanzapine Nano-Particles: In Vitro Characterization and in Vivo Evaluation, AAPS PharmSciTech (2016)
163. Enhanced Cytotoxicity to Cancer Cells by Codelivery and Controlled Release of Paclitaxel-Loaded Sirolimus-Conjugated Albumin Nanoparticles, Chemical Biology and Drug Design (2016)
164. Erratum: Drying of a Plasmid Containing Formulation: Chitosan As a Protecting Agent (Daru Journal of Pharmaceutical Sciences) (2016) 24 (11) Doi: 10.1186/2008-2231-20-29), DARU# Journal of Pharmaceutical Sciences (2016)
165. Fabrication and Biological Evaluation of Chitosan Coated Hyaluronic Acid-Docetaxel Conjugate Nanoparticles in Cd44+ Cancer Cells, DARU# Journal of Pharmaceutical Sciences (2016)
166. Hynic a Bifunctional Prosthetic Group for the Labelling of Peptides With 99Mtc and 18Fdg, Journal of Radioanalytical and Nuclear Chemistry (2016)
167. Laccase-Catalyzed Treatment of Ketoconazole, Identification of Biotransformed Metabolites, Determination of Kinetic Parameters, and Evaluation of Micro-Toxicity, Journal of Molecular Catalysis B: Enzymatic (2016)
168. Methylated 4-N,N Dimethyl Aminobenzyl N,O Carboxymethyl Chitosan As a New Chitosan Derivative: Synthesis, Characterization, Cytotoxicity and Antibacterial Activity, Carbohydrate Polymers (2016)
169. Nimodipine-Loaded Pluronic® Block Copolymer Micelles: Preparation, Characterization, In-Vitro and In-Vivo Studies, Iranian Journal of Pharmaceutical Research (2016)
170. Photocatalytic Removal of Doxycycline From Aqueous Solution Using Zno Nano-Particles: A Comparison Between Uv-C and Visible Light, Water Science and Technology (2016)
171. Preparation and Optimization of N-Trimethyl-O-Carboxymethyl Chitosan Nanoparticles for Delivery of Low-Molecular-Weight Heparin, Pharmaceutical Development and Technology (2016)
172. Preparation of 1-Fluoro-4-Methyl-9H-[Carbonyl-14C]Thioxanthen-9-One and Amine Derivatives, Journal of Labelled Compounds and Radiopharmaceuticals (2016)
173. Preparation of a Carbon-14 Analog of 2-[2-(4-(Dibenzo[B, F][1,4]Thiazepin-11-Yl)Piperazin-1-Yl)Ethoxy]Ethanol, Radiochemistry (2016)
174. Preparation of Diaminedicarboxyplatinum (Ii) Functionalized Single-Wall Carbon Nanotube Via Bingel Reaction As a Novel Cytotoxic Agent, Iranian Journal of Pharmaceutical Research (2016)
175. Preparation of Hydrogel Embedded Polymer-Growth Factor Conjugated Nanoparticles As a Diabetic Wound Dressing, Drug Development and Industrial Pharmacy (2016)
176. Self Assembled Hyaluronic Acid Nanoparticles As a Potential Carrier for Targeting the Inflamed Intestinal Mucosa, Carbohydrate Polymers (2016)
177. Synthesis of 11-14C-Quetiapine, 11-14C-Isoclotiapine and 10-(4-Methylpiperazin-1-Yl)Pyrido[4,3-B][1,4]Benzothiazepine[10-14C], Journal of Radioanalytical and Nuclear Chemistry (2016)
178. Synthesis of 2-(Methylsulfonyl)-5-(4-(Methylsulfonyl) Phenyl)-4-Phenyl-1H-[5-14C]Imidazole, a Selective Cox-2 Inhibitor, Via Asymmetrical Benzoins, Journal of Labelled Compounds and Radiopharmaceuticals (2016)
179. Synthesis of a Carbon-14 Analog of 8-Chloro-11- (4-Methyl-1-Piperazinyl)-11-[14C]-5H-Dibenzo[B,E][1,4]Diazepine (Clozapine) Using Microwave Irradiation, Radiochemistry (2016)
180. Synthesis of the Olanzapine Labeled by Carbon-14, Journal of Labelled Compounds and Radiopharmaceuticals (2016)
181. Synthesis, Conformational Assignment, and Anti-Inflammatory Activities of N-Arylidene-2-(4-Chloro-2-(2-Substituted Phenoxy)Phenyl)Acetic Acid Hydrazides, Medicinal Chemistry Research (2016)
182. Synthesis, Molecular Docking Study, and Cytotoxic Activity of 1,3,5-Triaryl Pyrazole Derivatives, Letters in Drug Design and Discovery (2016)
183. Synthesis, Molecular Docking Study, and Cytotoxic Activity of 3,4-Diaryl-5-(4-Pyridinyl)-1,2,4-Oxadiazole, Medicinal Chemistry (2016)
184. Synthesis, Radiolabeling, and Biological Evaluation of Peptide Likkpf Functionalized With Hynic As Apoptosis Imaging Agent, Iranian Journal of Pharmaceutical Research (2016)
185. Two Cox-2 Inhibitors Induce Apoptosis in Human Erythroleukemia K562cells by Modulating Nf-Κb and Fhc Pathways, DARU# Journal of Pharmaceutical Sciences (2016)
186. Vigna Radiata As a New Source for Biotransformation of Hydroquinone to Arbutin, Pharmaceutical Sciences (2016)
187. Anticonvulsant Activity of 1,2,4-Triazine Derivatives With Pyridyl Side Chain: Synthesis, Biological, and Computational Study, Medicinal Chemistry Research (2015)
188. Apoptotic Effects of Two Cox-2 Inhibitors on Breast Adenocarcinoma Cells Through Cox-2 Independent Pathway, Journal of Cellular Biochemistry (2015)
189. Cationic Albumin-Conjugated Chelating Agent As a Novel Brain Drug Delivery System in Neurodegeneration, Chemical Biology and Drug Design (2015)
190. Chitosan Polyplex Nanoparticle Vector for Mir-145 Expression in Mcf-7: Optimization by Design of Experiment, International Journal of Biological Macromolecules (2015)
191. Comparative Study of in Vitro Prooxidative Properties and Genotoxicity Induced by Aflatoxin B1 and Its Laccase-Mediated Detoxification Products, Chemosphere (2015)
192. Design, Synthesis and Evaluation of Antitubercular Activity of Novel Dihydropyridine Containing Imidazolyl Substituent, Iranian Journal of Pharmaceutical Research (2015)
193. Development of Acid-Resistant Alginate/Trimethyl Chitosan Nanoparticles Containing Cationic Β-Cyclodextrin Polymers for Insulin Oral Delivery, AAPS PharmSciTech (2015)
194. Enhanced Cellular Cytotoxicity and Antibacterial Activity of 18-Β-Glycyrrhetinic Acid by Albumin-Conjugated Plga Nanoparticles, Drug Research (2015)
195. Improved Anticancer Delivery of Paclitaxel by Albumin Surface Modification of Plga Nanoparticles, DARU# Journal of Pharmaceutical Sciences (2015)
196. Isolation and Structural Characterization of Coryxin, a Novel Cyclic Lipopeptide From Corynebacterium Xerosis Ns5 Having Emulsifying and Anti-Biofilm Activity, Colloids and Surfaces B: Biointerfaces (2015)
197. Phytochemical Investigation and Antifungal Activity of Daucus Littoralis Smith Sub Sp. Hyrcanicus Rech.F, Research Journal of Phytochemistry (2015)
198. Polymeric Micelles of Peg-Pla Copolymer As a Carrier for Salinomycin Against Gemcitabine-Resistant Pancreatic Cancer, Pharmaceutical Research (2015)
199. Preparation and Antibacterial Activity Evaluation of 18-Β-Glycyrrhetinic Acid Loaded Plga Nanoparticles, Iranian Journal of Pharmaceutical Research (2015)
200. Protein Corona Hampers Targeting Potential of Muc1 Aptamer Functionalized Sn-38 Core-Shell Nanoparticles, International Journal of Pharmaceutics (2015)
201. Synthesis and Anticancer Activity of 1,3,5-Triaryl-1H-Pyrazole, Letters in Drug Design and Discovery (2015)
202. Synthesis and Biological Evaluation of 5-Benzylidenerhodanine-3-Acetic Acid Derivatives As Ache and 15-Lox Inhibitors, Journal of Enzyme Inhibition and Medicinal Chemistry (2015)
203. Synthesis and Evaluation of Anti-Inflammatory and Analgesic Activities of New 1,2,4-Triazole Derivatives, Medicinal Chemistry (2015)
204. The Neuroprotective Effect of a Triazine Derivative in an Alzheimer’S Rat Model, Acta Medica Iranica (2015)